SDU
Denmark
Work
University of Southern Denmark
|Professor
Denmark
→
Education
The Royal Danish School of Pharmacy
Denmark
→
Ph.D.
The Royal Danish School of Pharmacy
Denmark
→
M.Sc. (Pharm)
Publications
Formulation Approaches for COVID-19 Vaccines
Nanotherapeutics for Infectious Diseases
book-chapter
Fragment-Based Screening Identifies Novel Non-Amino Acid Inhibitors of the Sodium-Coupled Neutral Amino Acid Transporter SNAT2
Pharmaceutical Research
journal-article
Fragment-Based Screening Identifies Novel Non-Amino Acid Inhibitors of the Sodium-Coupled Neutral Amino Acid Transporter SNAT2
Pharmaceutical Research
journal-article
Linker and Head-Group Exploration of Anti-MRSA Triaromatic Pleuromutilins
Journal of Medicinal Chemistry
journal-article
The oral bioavailability of a pleuromutilin antibiotic candidate is increased after co-administration with the CYP3A4 inhibitor ritonavir and the P-gp inhibitor zosuquidar formulated as amorphous solid dispersions
International Journal of Pharmaceutics
journal-article
Screening of a fragment-based library uncovers novel scaffolds for inhibitors of the sodium-coupled neutral amino acid transporter SNAT2
13th Uppsala University Symposium, 23/01/2025
conference-poster
Non-Steroidal Anti-Inflammatory Drugs Are Inhibitors of the Intestinal Proton-Coupled Amino Acid Transporter (PAT1): Ibuprofen and Diclofenac Are Non-Translocated Inhibitors
Pharmaceutics
journal-article
Non-Steroidal Anti-Inflammatory Drugs Are Inhibitors of the Intestinal Proton-Coupled Amino Acid Transporter (PAT1): Ibuprofen and Diclofenac Are Non-Translocated Inhibitors
Pharmaceutics
journal-article
Exploring Amino Acid Transporters as Therapeutic Targets for Cancer: An Examination of Inhibitor Structures, Selectivity Issues, and Discovery Approaches
Pharmaceutics
journal-article
The infectious capacity of Enterococcus faecalis, Staphylococcus aureus, and Staphylococcus saprophyticus in a porcine model of urinary tract infection
APMIS
journal-article
Structure-activity relationship of amino acid analogs to probe the binding pocket of sodium-coupled neutral amino acid transporter SNAT2
Amino Acids
journal-article
Digestion of surfactants does not affect their ability to inhibit P-gp-mediated transport in vitro
International Journal of Pharmaceutics
journal-article
Co-release of paclitaxel and encequidar from amorphous solid dispersions increase oral paclitaxel bioavailability in rats
International Journal of Pharmaceutics
journal-article
Hit-to-Lead Identification and Validation of a Triaromatic Pleuromutilin Antibiotic Candidate
Journal of Medicinal Chemistry
journal-article
Exploring Amino Acid Transporters as Therapeutic Targets for Cancer: An Examination of Inhibitor Structures, Selectivity Issues, and Discovery Approaches
Pharmaceutics
journal-article
Investigations of potential non-amino acid SNAT2 inhibitors.
Frontiers in Pharmacology
journal-article
Phloretin inhibits glucose transport and reduces inflammation in human retinal pigment epithelial cells
Molecular and Cellular Biochemistry
journal-article
Structure-based discovery of novel P-glycoprotein inhibitors targeting the nucleotide binding domains
Scientific Reports
journal-article
Probing the Substrate Binding Site of SNAT2 With Amino Acid Analogues: A Structure-Activity Relationship Study
RESOLUTE Conference, Wien, Austria, 27/09/2023
conference-poster
Increased bioavailability of a P-gp substrate
International Journal of Pharmaceutics
journal-article
Combinational Inhibition of P-Glycoprotein-Mediated Etoposide Transport by Zosuquidar and Polysorbate 20
Pharmaceutics
journal-article
Combinational Inhibition of P-Glycoprotein-Mediated Etoposide Transport by Zosuquidar and Polysorbate 20
Pharmaceutics
journal-article
Recent Advances in Photothermal Therapies Against Cancer and the Role of Membrane Transporter Modulators on the Efficacy of This Approach
Technology in Cancer Research and Treatment
journal-article
Molecular Networks and Macromolecular Molar Mass Distributions for Preliminary Characterization of Danish Craft Beers
Beverages
journal-article
In vitro and ex vivo evaluation of bilayered effervescent microenvironmental pH modifying buccal films with saquinavir
Journal of Drug Delivery Science and Technology
journal-article
SNAT2 is responsible for hyperosmotic induced sarcosine and glycine uptake in human prostate PC-3 cells
Pflügers Archiv - European Journal of Physiology
journal-article
P-glycoprotein-mediated transport in a mucus-supplemented Caco-2 cell model in the presence of different surfactants
International Journal of Pharmaceutics
journal-article
Mechanism behind Polysorbates’ Inhibitory Effect on P-Glycoprotein
Molecular Pharmaceutics
journal-article
Mechanism behind polysorbates' inhibitory effect on P-glycoprotein
Molecular Pharmaceutics
journal-article
Molecular Networks and Macromolecular Molar Mass Distributions for Preliminary Characterization of Danish Craft Beers
Beverages
journal-article
Oral etoposide and zosuquidar bioavailability in rats: Effect of co-administration and in vitro-in vivo correlation of P-glycoprotein inhibition
International Journal of Pharmaceutics: X
journal-article
Corrigendum to 'Is Oral Absorption of Vigabatrin Carrier-mediated?' [European Journal of Pharmaceutical Sciences 69 (2015) 10-18]
European Journal of Pharmaceutical Sciences
other
Exploration of in vitro drug release testing methods for saquinavir microenvironmental pH modifying buccal films
European Journal of Pharmaceutical Sciences
journal-article
Exploration of in vitro drug release testing methods for saquinavir microenvironmental pH modifying buccal films
European Journal of Pharmaceutical Sciences
journal-article
Inhibitory effects of 17-α-ethinyl-estradiol and 17-β-estradiol on transport via the intestinal proton-coupled amino acid transporter (PAT1) investigated In vitro and in vivo
Journal of Pharmaceutical Sciences
journal-article
BeerMIMS
European Journal of Mass Spectrometry
journal-article
Acamprosate Is a Substrate of the Human Organic Anion Transporter (OAT) 1 without OAT3 Inhibitory Properties
Pharmaceutics
journal-article
Evaluation of P-glycoprotein efflux activity and cellular toxicity in MDCKII MDR1 cells in a one-pot assay
Nordic POP Annual meeting 2020 , Copenhagen , Denmark, 07/01/2020
conference-poster
Zosuquidar alters etoposide permeability across Caco-2 cell monolayers by P-glycoprotein inhibition in a concentration-dependent manner
Nordic POP Annual meeting 2020 , Copenhagen , Denmark, 07/01/2020
conference-poster
Discovery of a Potent Adenine-Benzyltriazolo-Pleuromutilin Conjugate with Pronounced Antibacterial Activity against MRSA
Journal of Medicinal Chemistry
journal-article
Microenvironmental pH modifying films for buccal delivery of saquinavir
International Journal of Pharmaceutics
journal-article
High-dose etoposide formulations do not saturate intestinal P-glycoprotein
International Journal of Pharmaceutics
journal-article
Acamprosate Is a Substrate of the Human Organic Anion Transporter (OAT) 1 without OAT3 Inhibitory Properties: Implications for Renal Acamprosate Secretion and Drug–Drug Interactions
Pharmaceutics
journal-article
Acamprosate Is a Substrate of the Human Organic Anion Transporter (OAT) 1 without OAT3 Inhibitory Properties: Implications for Renal Acamprosate Secretion and Drug–Drug Interactions
Pharmaceutics
journal-article
Etoposide transport in MDCKII-MRP2 cells is unaffected by P-gp expression and commonly used pharmaceutical excipients
Nordic POP 1st Annual Meeting, Oslo, Norway, 14/01/2019
conference-output
Transcriptome analysis identifies activated signaling pathways and regulated ABC transporters and solute carriers after hyperosmotic stress in renal MDCK I cells
Genomics
journal-article
Transcriptome analysis identifies activated signaling pathways and regulated ABC transporters and solute carriers after hyperosmotic stress in renal MDCK I cells
Genomics
journal-article
The permeation of acamprosate is predominantly caused by paracellular diffusion across Caco-2 cell monolayers
Molecular Pharmaceutics
journal-article
The Permeation of Acamprosate Is Predominantly Caused by Paracellular Diffusion across Caco-2 Cell Monolayers: A Paracellular Modeling Approach
Molecular Pharmaceutics
journal-article
Montmorillonite-surfactant hybrid particles for modulating intestinal P-glycoprotein-mediated transport
International Journal of Pharmaceutics
journal-article
Montmorillonite-surfactant hybrid particles for modulating intestinal P-glycoprotein-mediated transport
International Journal of Pharmaceutics
journal-article
Nonionic surfactants modulate the transport activity of ATP-binding cassette (ABC) transporters and solute carriers (SLC)
International Journal of Pharmaceutics
journal-article
MRP2-mediated transport of etoposide in MDCKII MRP2 cells is unaffected by commonly used non-ionic surfactants
International Journal of Pharmaceutics
journal-article
Nfat5 is involved in the hyperosmotic regulation of Tmem184b: a putative modulator of ibuprofen transport in renal MDCK I cells
FEBS Open Bio
journal-article
Nfat5 is involved in the hyperosmotic regulation of Tmem184b
FEBS Open Bio
journal-article
Acamprosate is an inhibitor of the renal organic anion transporter (OAT) 1
Nordic POP 1st Annual Meeting, Oslo, Norway, 14/01/2019
conference-output
Montmorillonite-surfactant hybrid particles for modulation of intestinal P-glycoprotein mediated transport
Nordic POP 1st Annual Meeting, Oslo, Norway, 14/01/2019
conference-poster
Amino acid transport in prostate PC-3 cells
Nordic POP 1st Annual Meeting, Oslo, Norway, 14/01/2019
conference-output
Acamprosate permeability across Caco-2 cell monolayer is predominantly paracellular
Northern Pharma Network Meeting & POP Kick off-Meeting Conference 2018, Odense, Odense, Denmark, 29/01/2018
conference-output
Nonionic surfactants increase digoxin absorption in Caco-2 and MDCKII MDR1 cells
International Journal of Pharmaceutics
journal-article
How is sarcosine transported into prostate PC‐3 cells?
The Danish Chemical Society Annual Meeting 2018
, Odense, Denmark, 23/08/2018
conference-poster
Hyperosmolality regulates mRNA expression of membrane transporters in renal MDCK I cells
Northern Pharma Network Meeting & POP Kick off-Meeting Conference, Odense, Denmark, 29/01/2018
conference-poster
Nonionic surfactants alter calcein-AM efflux in MDCKII MDR1 cells
Northern Pharma Network Meeting & POP Kick off-Meeting Conference 2018, Odense, Odense, Denmark, 29/01/2018
conference-poster
Polysorbate 20 alters the oral bioavailability of etoposide in wild type and mdr1a deficient Sprague-Dawley rats
International Journal of Pharmaceutics
journal-article
Glutamate Transporters in the Blood-Brain Barrier
Glial Amino Acid Transporters
book-chapter
Transport and metabolism of l‑glutamate in brain capillary endothelial cells and astrocytes
Fluids and Barriers of the CNS
conference-abstract
Oral and intravenous pharmacokinetics of taurine in sprague-dawley rats: the influence of dose and the possible involvement of the proton-coupled amino acid transporter, PAT1, in oral taurine absorption
Physiological Reports
journal-article
Oral and intravenous pharmacokinetics of taurine in sprague-dawley rats
Physiological Reports
journal-article
SGLT1-Mediated Transport in Caco-2 Cells Is Highly Dependent on Cell Bank Origin.
Journal of pharmaceutical sciences
journal-article
SGLT1-mediated transport in Caco-2 cells is highly dependent on cell bank origin
Journal of Pharmaceutical Sciences
journal-article
Characterization of the L-glutamate clearance pathways across the blood-brain barrier and the effect of astrocytes in an in vitro blood-brain barrier model.
Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism
journal-article
Characterization of the L-glutamate clearance pathways across the blood-brain barrier and the effect of astrocytes in an in vitro blood-brain barrier model
Journal of Cerebral Blood Flow & Metabolism
journal-article
Glutamate Transporters in the Blood-Brain Barrier.
Advances in neurobiology
journal-article
A Transporter of Ibuprofen is Upregulated in MDCK I cells under Hyperosmotic Culture Conditions
Molecular Pharmaceutics
journal-article
Application of Cell Culture and Tissue Models for Assessing Drug Transport
Analytical Techniques in the Pharmaceutical Sciences
book-chapter
Hyperosmolality regulates transporters in renal MDCK I cells
The Annual Meeting of the Danish Chemical Society, Odense, Denmark, 09/06/2016
conference-poster
Ibuprofen transport in renal cell cultures: Characterization of an ibuprofen transporter upregulated by hyperosmolarity
MedChemComm
journal-article
Ibuprofen transport in renal cell cultures: characterization of an ibuprofen transporter upregulated by hyperosmolarity
MedChemComm
journal-article
Ibuprofen transport in renal cell cultures
MedChemComm
journal-article
PAT1 contributes to the absorption of taurine in vivo
The Annual Meeting of the Danish Chemical Society, Odense, Denmark, 09/06/2016
conference-poster
Tween 20 increases intestinal transport of doxorubicin in vitro but not in vivo
International Journal of Pharmaceutics
journal-article
Tween 20 increase absorptive digoxin transport in MDCKII-MDR1 cells
The Annual Meeting of the Danish Chemical Society, Odense, Denmark, 09/06/2016
conference-poster
Polysorbate 20 increases oral absorption of digoxin in wild-type Sprague Dawley rats, but not in mdr1a(-/-) Sprague Dawley rats
International Journal of Pharmaceutics
journal-article
Polysorbate 20 increases oral absorption of digoxin in wild-type Sprague Dawley rats, but not in mdr1a(-/-) Sprague Dawley rats
International Journal of Pharmaceutics
journal-article
Tween 20 increases intestinal transport of doxorubicin in vitro but not in vivo
International Journal of Pharmaceutics
journal-article
Interaction of GABA-mimetics with the taurine transporter (TauT, Slc6a6) in hyperosmotic treated Caco-2, LLC-PK1 and rat renal SKPT cells
European Journal of Pharmaceutical Sciences
journal-article
Interaction of GABA-mimetics with the taurine transporter (TauT, Slc6a6) in hyperosmotic treated Caco-2, LLC-PK1 and rat renal SKPT cells
European Journal of Pharmaceutical Sciences
journal-article
Interaction of GABA-mimetics with the taurine transporter (TauT, Slc6a6) in hyperosmotic treated caco-2, LLC-PK1 and rat renal SKPT cells
European Journal of Pharmaceutical Sciences
journal-article
17-β-estradiol and ethinyl-estradiol inhibit PAT1-mediated taurine transport in Caco-2 cells, but doesn’t alter the pharmacokinetic profile in vivo
The Annual Meeting of the Danish Chemical Society, Odense, Denmark, 09/06/2016
conference-poster
A transporter of ibuprofen is upregulated in MDCK i cells under hyperosmotic culture conditions
Molecular Pharmaceutics
journal-article
Is oral absorption of vigabatrin carrier-mediated?
European Journal of Pharmaceutical Sciences
journal-article
Estradiol and ethinyl-estradiol decrease proline uptake and transport in intestinal Caco-2 cells
Amino Acids
conference-abstract
Is oral absorption of vigabatrin carrier-mediated?
European Journal of Pharmaceutical Sciences
journal-article
The anti-epileptic drug substance vigabatrin inhibits transport via the taurine transporter (TauT, SLC6A6) in SKPT cells
Amino Acids
conference-abstract
In vivo and In vitro Evaluations of Intestinal Gabapentin Absorption
Pharmaceutical Research
journal-article
IN VITRO MEMBRANE PERMEATION STUDIES AND IN VIVO ANTINOCICEPTION OF GLYCOSYLATED Dmt1-DALDA ANALOGUES
33rd European Peptide Society Symposium, Sofia, Bulgaria, 31/08/2014
conference-presentation
Efflux transporter expression in a tight in vitro model of the blood brain barrier
Cold Spring Harbor Conference, Cold Spring Harbor, United States, 10/12/2014
conference-output
Transport pathways mediating blood-to-brain L-glutamate efflux
Cold Spring Harbor Conference, Cold Spring Harbor, United States, 10/12/2014
conference-output
Glutamate Efflux at the Blood-Brain Barrier
Archives of Medical Research
journal-article
The anti-epileptic drug substance vigabatrin inhibits taurine transport in intestinal and renal cell culture models.
journal-article
The anti-epileptic drug substance vigabatrin inhibits taurine transport in intestinal and renal cell culture models
International Journal of Pharmaceutics
journal-article
The anti-epileptic drug substance vigabatrin inhibits taurine transport in intestinal and renal cell culture models
International Journal of Pharmaceutics
journal-article
A Tight Blood-Brain Barrier Model Displays Brain-to-Blood Efflux of Substrates for the ABC-Transporters, P-gp, BCRP and MRP-1
Signal Transduction in The Blood-Brain Barriers, Potsdam, Germany, 13/09/2012
conference-output
An electrically tight in vitro blood-brain barrier model displays net brain-to-blood efflux of substrates for the ABC transporters, P-gp, Bcrp and Mrp-1
AAPS Journal
journal-article
An Electrically Tight In Vitro Blood-Brain Barrier Model Displays Net Brain-to-Blood Efflux of Substrates for the ABC Transporters, P-gp, Bcrp and Mrp-1
The AAPS Journal
journal-article
In vivo and In vitro Evaluations of Intestinal Gabapentin Absorption: Effect of Dose and Inhibitors on Carrier-Mediated Transport.
journal-article
Pharmacokinetic aspects of the anti-epileptic drug substance vigabatrin: Focus on transporter interactions
Therapeutic Delivery
journal-article
The absorptive flux of the anti-epileptic drug substance vigabatrin is carrier-mediated across Caco-2 cell monolayers
European Journal of Pharmaceutical Sciences
journal-article
IN VITRO MEMBRANE PERMEATION STUDIES AND IN VIVO ANTINOCICEPTION OF GLYCOSYLATED Dmt1-DALDA ANALOGUES
33rd European Peptide Society Symposium, Sofia, Bulgaria, 31/08/2014
conference-output
Intestinal absorption of the antiepileptic drug substance vigabatrin in Gottingen mini-pigs is unaffected by co-administration of amino acids.
journal-article
Intestinal absorption of the antiepileptic drug substance vigabatrin in Göttingen mini-pigs is unaffected by co-administration of amino acids
International Journal of Pharmaceutics
journal-article
Intestinal absorption of the antiepileptic drug substance vigabatrin in Göttingen mini-pigs is unaffected by co-administration of amino acids
International Journal of Pharmaceutics
journal-article
Design of prodrugs targeting the intestinal di/tri‐peptide transporter hPEPT1 (SLC15A1
Meet the Experts: Transporter Conference- 2014, Budapest, Hungary, 02/04/2014
conference-output
In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt(1)-DALDA Analogues.
journal-article
In vitro membrane permeation studies and in vivo antinociception of glycosylated Dmt1-DALDA analogues
ACS Medicinal Chemistry Letters
journal-article
In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt1-DALDA Analogues
ACS Medicinal Chemistry Letters
journal-article
Intestinal absorption of the antiepileptic drug substance vigabatrin is altered by infant formula in vitro and in vivo
Pharmacology Research & Perspectives
journal-article
PAT1 (SLC36A1) shows nuclear localization and affects growth of smooth muscle cells from rats.
journal-article
PAT1 (SLC36A1) shows nuclear localization and affects growth of smooth muscle cells from rats
American Journal of Physiology - Endocrinology and Metabolism
journal-article
PAT1 (SLC36A1) shows nuclear localization and affects growth of smooth muscle cells from rats
American Journal of Physiology: Endocrinology and Metabolism
journal-article
An electrically tight in vitro blood-brain barrier model displays net brain-to-blood efflux of substrates for the ABC transporters, P-gp, Bcrp and Mrp-1.
journal-article
The absorptive flux of the anti-epileptic drug substance vigabatrin is carrier-mediated across Caco-2 cell monolayers.
journal-article
Pharmacokinetic aspects of the anti-epileptic drug substance vigabatrin
Therapeutic Delivery
journal-article
The absorptive flux of the anti-epileptic drug substance vigabatrin is carrier-mediated across Caco-2 cell monolayers
European Journal of Pharmaceutical Sciences
journal-article
Vigabatrin absorption is mediated via the proton-coupled amino acid transporter PAT1 – in vitro and in vivo
conference-poster
In vivo and in vitro evaluations of intestinal gabapentin absorption: Effect of dose and inhibitors on carrier-mediated transport
Pharmaceutical Research
journal-article
Sertraline inhibits the transport of PAT1 substrates in vivo and in vitro.
journal-article
Sertraline inhibits the transport of PAT1 substrates in vivo and in vitro
British Journal of Pharmacology
journal-article
Sertraline inhibits the transport of PAT1 substrates in vivo and in vitro
British Journal of Pharmacology
journal-article
Basolateral glycylsarcosine (Gly-Sar) transport in Caco-2 cell monolayers is pH dependent.
journal-article
Basolateral glycylsarcosine (Gly-Sar) transport in Caco-2 cell monolayers is pH dependent
Journal of Pharmacy and Pharmacology
journal-article
Basolateral glycylsarcosine (Gly-Sar) transport in Caco-2 cell monolayers is pH dependent
Journal of Pharmacy and Pharmacology
journal-article
PAT1-inhibitors reduce oral absorption rate of vigabatrin in rats
PAGE 2013, Glasgow, United Kingdom, 11/06/2013
conference-poster
Excitatory amino acid transporter-1 (EAAT1) is the main transporter responsible for abluminal uptake of L-glutamate in bovine brain endothelial cells
45 Sandbjerg Meeting on Membrane Transport, Sønderborg, Denmark, 27/05/2013
conference-output
Cellemodel af blodhjernebarrieren kan mindske brugen af forsøgsdyr
Lægemiddelforskning
journal-article
Current status of rational design of prodrugs targeting the intestinal di/tri-peptide transporter hPEPT1 (SLC15A1)
Journal of Drug Delivery Science and Technology
journal-article
Current status of rational design of prodrugs targeting the intestinal di/tri-peptide transporter hPEPT1 (SLC15A1)
Journal of Drug Delivery Science and Technology
journal-article
Membrane Transporters in ADME
Transporters in Drug Development
book-chapter
Potential involvement of the proton-coupled amino acid transporter PAT1 (SLC36A1) in the delivery of pharmaceutical agents
Journal of Drug Delivery Science and Technology
journal-article
Potential involvement of the proton-coupled amino acid transporter PAT1 (SLC36A1) in the delivery of pharmaceutical agents
Journal of Drug Delivery Science and Technology
journal-article
In-vitro models of the blood brain barrier
44th Sandbjerg Meeting on Membrane Transport, Sandbjerg, Denmark, 14/05/2012
conference-output
Kostens sammensætning kan påvirke optagelsen af lægemiddelstoffer
Lægemiddelforskning
journal-article
The proton-coupled amino acid transporter hPAT1 is the main transporter involved in vigabatrin uptake in intestinal Caco-2 cells
conference-poster
Function and expression of the proton-coupled amino acid transporter PAT1 along the rat gastrointestinal tract: implications for intestinal absorption of gaboxadol.
journal-article
Function and expression of the proton-coupled amino acid transporter PAT1 along the rat gastrointestinal tract: Implications for intestinal absorption of gaboxadol
British Journal of Pharmacology
journal-article
Function and expression of the proton-coupled amino acid transporter Slc36a1 along the rat gastrointestinal tract
British Journal of Pharmacology
journal-article
In vitro evidence for the brain glutamate efflux hypothesis: brain endothelial cells co-cultured with astrocytes display a polarized brain-to-blood transport of glutamate
Signal Transduction in The Blood-Brain Barriers, Potsdam, Germany, 13/09/2012
conference-output
Intestinal drug transport via the proton-coupled amino acid transporter PAT1 (SLC36A1) is inhibited by Gly-X(aa) dipeptides.
journal-article
Intestinal drug transport via the proton-coupled amino acid transporter PAT1 (SLC36A1) is inhibited by gly-Xaa dipeptides
Molecular Pharmaceutics
journal-article
Intestinal drug transport via the proton-coupled amino acid transporter PAT1 (SLC36A1) is inhibited by Gly-X(aa) dipeptides
Molecular Pharmaceutics
journal-article
Carrier-mediated γ-aminobutyric acid transport across the basolateral membrane of human intestinal Caco-2 cell monolayers.
journal-article
Carrier-mediated γ-aminobutyric acid transport across the basolateral membrane of human intestinal Caco-2 cell monolayers
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
Carrier-mediated ¿-aminobutyric acid transport across the basolateral membrane of human intestinal Caco-2 cell monolayers
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
In vitro evidence for the brain glutamate efflux hypothesis: brain endothelial cells cocultured with astrocytes display a polarized brain-to-blood transport of glutamate.
journal-article
In vitro evidence for the brain glutamate efflux hypothesis: Brain endothelial cells cocultured with astrocytes display a polarized brain-to-blood transport of glutamate
GLIA
journal-article
In vitro evidence for the brain glutamate efflux hypothesis
Glia
journal-article
Rectal absorption of vigabatrin, a substrate of the proton coupled amino acid transporter (PAT1, Slc36a1), in rats.
journal-article
Rectal absorption of vigabatrin, a substrate of the proton coupled amino acid transporter (PAT1, Slc36a1), in rats
Pharmaceutical Research
journal-article
Rectal absorption of vigabatrin, a substrate of the proton coupled amino acid transporter (PATI, Slc36ai) in rats
Pharmaceutical Research
journal-article
Glutamate efflux from brain to blood - Studies in an in vitro blood-brain barrier model
44'th Sandbjerg Meeting on Membrane Transport, Sønderborg, Denmark, 14/05/2012
conference-output
Identification and Characterization of a Novel Nontranslated Sequence Variant of the Human Intestinal Di-/Tripeptide Transporter, hPEPT1.
journal-article
Identification and characterization of a novel nontranslated sequence variant of the human intestinal Di-/Tripeptide transporter, hPEPT1
International Journal of Peptides
journal-article
Identification and Characterization of a Novel Nontranslated Sequence Variant of the Human Intestinal Di-/Tripeptide Transporter, hPEPT1
International Journal of Peptides
journal-article
Gaboxadol has affinity for the proton-coupled amino acid transporter 1, SLC36A1(hPAT1)-A modelling approach to determine IC50 values of the three ionic species of gaboxadol
European Journal of Pharmaceutical Sciences
journal-article
Transport af lægemiddelstoffer gennem vævsbarrier
Bioteknologi - en temabog
book-chapter
The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1.
journal-article
The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1
Bioorganic and Medicinal Chemistry Letters
journal-article
The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1
Bioorganic & Medicinal Chemistry Letters
journal-article
Calu-3 cells grown under AIC and LCC conditions: implications for dipeptide uptake and transepithelial transport of substances.
journal-article
Calu-3 cells grown under AIC and LCC conditions: Implications for dipeptide uptake and transepithelial transport of substances
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
Calu-3 cells grown under AIC and LCC conditions
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
Affinity and translocation relationships via hPEPT1 of H-X aa-Ser-OH dipeptides: evaluation of H-Phe-Ser-OH as a pro-moiety for ibuprofen and benzoic acid prodrugs.
journal-article
Affinity and translocation relationships via hPEPT1 of H-X aa-Ser-OH dipeptides: Evaluation of H-Phe-Ser-OH as a pro-moiety for ibuprofen and benzoic acid prodrugs
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
Affinity and translocation relationships via hPEPT1 of H-Xaa-Ser-OH dipeptides
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
Gaboxadol has affinity for the proton-coupled amino acid transporter 1, SLC36A1 (hPAT1)--A modelling approach to determine IC(50) values of the three ionic species of gaboxadol.
journal-article
Gaboxadol has affinity for the proton-coupled amino acid transporter 1, SLC36A1 (hPAT1) - A modelling approach to determine IC50 values of the three ionic species of gaboxadol
European Journal of Pharmaceutical Sciences
journal-article
Stoftransport af lægemiddelstoffer gennem vævsbarrierer.
Bioteknologi – en temabog.
book-chapter
A quantitative structure-activity relationship for translocation of tripeptides via the human proton-coupled peptide transporter, hPEPT1 (SLC15A1)
AAPS Journal
journal-article
Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): possible interactions between hPEPT1 substrates and ibuprofen.
journal-article
Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): Possible interactions between hPEPT1 substrates and ibuprofen
British Journal of Pharmacology
journal-article
Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): possible interactions between hPEPT1 substrates and ibuprofen
British Journal of Pharmacology
journal-article
Paracellular tightness and claudin-5 expression is increased in the BCEC/astrocyte blood-brain barrier model by increasing media buffer capacity during growth.
journal-article
Paracellular tightness and claudin-5 expression is increased in the bcec/astrocyte blood-brain barrier model by increasing media buffer capacity during growth
AAPS Journal
journal-article
Paracellular tightness and claudin-5 expression is increased in the BCEC/Astrocyte blood-brain barrier model by increasing media buffer capacity during growth
The AAPS Journal
journal-article
The proton-coupled amino acid transporter, SLC36A1 (hPAT1), transports Gly-Gly, Gly-Sar and other Gly-Gly mimetics
British Journal of Pharmacology
journal-article
The proton-coupled amino acid transporter, SLC36A1 (hPAT1), transports Gly-Gly, Gly-Sar and other Gly-Gly mimetics
British Journal of Pharmacology
journal-article
A quantitative structure-activity relationship for translocation of tripeptides via the human proton-coupled peptide transporter, hPEPT1 (SLC15A1).
journal-article
A Quantitative Structure–Activity Relationship for Translocation of Tripeptides via the Human Proton-Coupled Peptide Transporter, hPEPT1 (SLC15A1)
The AAPS Journal
journal-article
Delta-aminolevulinic acid is a substrate for the amino acid transporter SLC36A1 (hPAT1).
journal-article
δ-Aminolevulinic acid is a substrate for the amino acid transporter SLC36A1 (hPAT1)
British Journal of Pharmacology
journal-article
d-Aminolevulinic acid is a substrate for the amino acid transporter SLC36A1 (hPAT1)
British Journal of Pharmacology
journal-article
Gly-Sar is a substrate for the human proton-coupled amino acid transporter, hPAT1 (SLC36A1)
Joint meeting of the Scandinavian and german physiological societies, Copenhagen, Denmark, 27/03/2010
conference-output
Ibuprofen is an inhibitor of hPEPT1: Implications for drug-drug interactions at the level of drug absorption
Joint meeting of the Scandinavian and german physiological societies, Copenhagen, Denmark, 27/03/2010
conference-output
mRNA expression and transport function of the proton-coupled amino acid transporter , PAT1, along the rat intestine
Joint meeting of the Scandinavian and german physiological societies, Copenhagen, Denmark, 27/03/2010
conference-output
5-Hydroxy-L-tryptophan alters gaboxadol pharmacokinetics in rats: involvement of PAT1 and rOat1 in gaboxadol absorption and elimination.
journal-article
5-Hydroxy-l-tryptophan alters gaboxadol pharmacokinetics in rats: Involvement of PAT1 and rOat1 in gaboxadol absorption and elimination
European Journal of Pharmaceutical Sciences
journal-article
5-Hydroxy-L-tryptohan alters gaboxadol pharmacokinetics in rats
European Journal of Pharmaceutical Sciences
journal-article
Absorptive transporters
Molecular Biopharmaceutics
book-chapter
Acid/base properties, solubility and distribution of drug candidates
Molecular Biopharmaceutics
book-chapter
Carrier-mediated transport kinetics
Molecular Biopharmaceutics
book-chapter
Claudin-5 mRNA expression and transendothelial electrical resistance (TEER) correlate in the BCEC/astrocyte blood-brain barrier model
2010 AAPS Annual Meeting and Exposition, New Orleans, United States, 14/11/2010
conference-output
Efflux transporters
Molecular Biopharmaceutics
book-chapter
GABA transport across the basolateral membrane of intestinal cells
Joint Meeting of the Scandinavian and German Physiological Societies, København, Denmark, 27/03/2010
conference-output
Gly-sar is a substrate for the human proton coupled amino acid trasporter 1, hPAT1 (SLC36A1)
Joint meeting of the Scandinavian and german physiological societies, Copenhagen, Denmark, 27/03/2010
conference-poster
Hjernens forsvarsmur kortlagt og kopieret
Lægemiddelforskning
journal-article
Ibuprofen is an inhibitor of hPEPT1: Implications for drug-drug interactions at the level of drug absorption
Ibuprofen is an inhibitor of hPEPT1: Implications for drug-drug interactions at the level of drug absorption, Copenhagen, Denmark, 27/03/2010
conference-poster
In vitro models for investigating the function of proton-coupled amino acid transporter 1 (PAT1, SLC36A19)
2010 AAPS Annual Meeting and Exposition, New Orleans, United States, 14/11/2010
conference-output
Introduction
Molecular biopharmaceutics
book-chapter
Introduction
Molecular Biopharmaceutics
book-chapter
Kinetics of decomposition in aqueous solution
Molecular Biopharmaceutics
book-chapter
Mechanisms of decomposition of drug candidates
Molecular Biopharmaceutics
book-chapter
Passive diffusion of drug substances
Molecular Biopharmaceutics
book-chapter
Structure and function of absorption barriers
Molecular Biopharmaceutics
book-chapter
The expression of Claudin-5 correlates with transendothelial electrical resistance (TEER) in BCEC/rat astrocyte blood-brain barrier models
Globalization of Pharmaceutics Education Network Meeting 2010, Chapel Hill, North Carolina, United States, 09/11/2010
conference-output
Transportes in gastrointestinal tract
Drug bioavailability
book-chapter
mRNA expression and transport function of the proton-coupled amino acid transporter, PAT1, along the rat intestine
Joint Meeting of the Scandinavian and German Physiological Societies, København, Denmark, 27/03/2010
conference-output
The proton-coupled amino acid transporter, SLC36A1 (hPAT1), transports Gly-Gly, Gly-Sar and other Gly-Gly mimetics.
journal-article
Gaboxadol bliver absorberet via en aminosyretransportør
Lægemiddelforskning
journal-article
Discovery of ligands for the human intestinal Di-/Tripeptide transporter (hPEPT1) using a QSAR-assisted virtual screening strategy.
journal-article
Discovery of ligands for the human intestinal Di-/tripeptide transporter (hPEPT1) using a QSAR-assisted virtual screening strategy
ChemMedChem
journal-article
Discovery of ligands for the human intestinal di-/tripeptide transporter (hPEPT1) using af QSAR-assisted virtual screening strategy
ChemMedChem
journal-article
Characterization of in-vitro blood-brain barrier models
BioMedical Transporters 2009, Bern, Switzerland, 09/08/2009
conference-output
Intestinal gaboxadol absorption via PAT1 (SLC36A1): modified absorption in vivo following co-administration of L-tryptophan.
journal-article
Intestinal gaboxadol absorption via PAT1 (SLC36A1): Modified absorption in vivo following co-administration of L-tryptophan
British Journal of Pharmacology
journal-article
Intestinal gaboxadol absorption via PAT1 (SLC36A1)
British Journal of Pharmacology
journal-article
Transport of Gaboxadol via hPAT1 and rOAT1 in the absence and presence of 5-HTP
36th Annual Meeting & Exposition of the controlled release society - Innovation in discovery, diagnostics, and delivery, Copenhagen, Denmark, 18/07/2009
conference-output
In vitro blood-brain barrier models
36th Annual Meeting & Exposition of the controlled release society - Innovation in discovery, diagnostics, and delivery, Copenhagen, Denmark, 18/07/2009
conference-output
Transporters in the gastrointestinal tract
Drug Bioavailability:
book-chapter
Modified absorption formulation of gaboxadol
patent
Peptide transporters in drug delivery; The human peptide transporter 1 (hPEPT1) translocates differently charged peptides in an electrogenic manner, indicating a varying proton coupling ration
41th Sandbjerg Meeting om Membrane Transport, Sønderborg, Denmark, 11/05/2009
conference-output
Dipeptide derivatives of AZT: synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity.
journal-article
Transport of amino acids and GABA analogues via the human proton-coupled amino acid transporter, hPAT1: characterization of conditions for affinity and transport experiments in Caco-2 cells.
journal-article
Transport of amino acids and GABA analogues via the human proton-coupled amino acid transporter, hPAT1: Characterization of conditions for affinity and transport experiments in Caco-2 cells
European Journal of Pharmaceutical Sciences
journal-article
Transport of amino acids and GABA analogues via the human proton-coupled amino acid transporter, hPAT1
European Journal of Pharmaceutical Sciences
journal-article
Dipeptide derivatives of AZT: Synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity
ChemMedChem
journal-article
Dipeptide derivatives of AZT
ChemMedChem
journal-article
hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3.
journal-article
hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3
Pflugers Archiv European Journal of Physiology
journal-article
hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3
Pflügers Archiv - European Journal of Physiology
journal-article
Cloning of the pig PEPT2 (pPEPT2) and characterization of the effects of epidermal growth factor (EGF) on pPEPT2-mediated peptide uptake in the renal porcine cell line LLC-PK1.
journal-article
Cloning of the pig PEPT2 (pPEPT2) and characterization of the effects of epidermal growth factor (EGF) on pPEPT2-mediated peptide uptake in the renal porcine cell line LLC-PK1
European Journal of Pharmaceutical Sciences
journal-article
Cloning of the pig PEPT2 (pPEPT2) and characterization of the effects of epidermal growth factor (EGF) on pPEPT2-mediated peptide uptake in the renal porcine cell line LLC-PK1
European Journal of Pharmaceutical Sciences
journal-article
Basolateral peptid etransport in the human intestinal cell line Caco-2 is proton-coupled
Globalization of Pharmaceutics Education Network Meeting 2008, Leuven, Belgium, 09/09/2008
conference-output
Design, synthesis, and evaluation of tripeptidic promoieties targeting the intestinal peptide transporter hPEPT1
ChemMedChem
journal-article
Design, synthesis, and evaluation of tripeptidic promoieties targeting the intestinal peptide transporter hPEPT1
ChemMedChem
journal-article
Proton-coupled basolateral dipeptide transport in a human intestinal cell line, Caco-2
3rd Pharmaceutical Sciences World Congress, Amsterdam, Netherlands, 22/04/2007
conference-output
The human proton-coupled amino acid transporter (hPAT1) is a transport system for GABA-like drugs
22007 Annual AAPS Meeting, San Diego, United States, 11/11/2007
conference-output
Design, synthesis, and evaluation of tripeptidic promoieties targeting the intestinal peptide transporter hPEPT1.
journal-article
Transportpeptider
Lægemiddelforskning
journal-article
Basolateral peptide transport in intestinal cells is pH dependent
39th Sandbjerg Meeting on Membrane Transport, Sandbjerg, Denmark, 16/05/2007
conference-output
Molekylær biofarmaci - når medicinen skyder genvej!
Lægemiddelforskning
journal-article
Optimization of a cell-based flourescent probe assay for measuring substrate translocation via the proton-coupled intestinal di/tri-peptide transporter hPEPT1
ULLA Summerschool 2007, Leiden, Netherlands, 29/06/2007
conference-output
Peptide Transporters in Drug Delivery
Joint meeting of the German and the Danish Pharmacological Societies, Copenhagen, Denmark, 21/06/2007
conference-output
In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1
European Journal of Pharmaceutical Sciences
journal-article
Carbonic anhydrase inhibitors: transepithelial transport of thioureido sulfonamide inhibitors of the cancer-associated isozyme IX is dependent on efflux transporters.
journal-article
Carbonic anhydrase imhibitors. Transepithelial transport of novel anticancer sulfonamide inhibitors of the cancer-associated isozyme CA IX is dependent on the p.gp efflux transporter
Bioorganic & Medicinal Chemistry Letters
journal-article
Development of a QSAR model for binding of tripeptides and tripeptidomimetics to the human intestinal di-/tripeptide transporter hPEPT1.
journal-article
Genetic variants of the human dipeptide transporter PEPT1
The Journal of Pharmacology and Experimental Therapeutics
journal-article
Genetic variants of the human dipeptide transporter PEPT1
Journal of Pharmacology and Experimental Therapeutics
journal-article
Development of a QSAR model for binding of tripeptides and tripeptidomimetics to the human intestinal di-/tripeptide transporter hPEPT1
Pharmaceutical Research
journal-article
Development of a QSAR model for binding of tripeptides and tripeptidomimetics to the human intestinal Di-/tripeptide transporter hPEPT1
Pharmaceutical Research
journal-article
Genetic variants of the human dipeptide transporter PEPT1.
journal-article
In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1.
journal-article
In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1
European Journal of Pharmaceutical Sciences
journal-article
Carbonic anhydrase inhibitors: Transepithelial transport of thioureido sulfonamide inhibitors of the cancer-associated isozyme IX is dependent on efflux transporters
Bioorganic and Medicinal Chemistry
journal-article
Carrier-mediated dipeptide transport in a human lung epithelial cell line, Calu-3
American Association of Pharmaceutical Scientists (AAPS) annual meeting and exhibition, San Antonio, United States, 12/11/2006
conference-output
Insulin increases peptide transport capacity in the proximal tubule kidney cell line SKPT0193-Cl.2.
American Association of Pharmaceutical Scientists (AAPS) annual meeting and exhibition, San Antonio, United States, 12/11/2006
conference-output
Proton dependent transport of amino acids in Caco-2 cells
Sandbjerg Meeting on Membrane Transport, Sandbjerg, Denmark, 31/05/2006
conference-output
Delivery aspects of small peptides and substrates for peptide transporters.
journal-article
Delivery aspects of small peptides and substrates for peptide transporters
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
Delivery aspects of small peptides and substrates for peptide transporters
European Journal of Pharmaceutics and Biopharmaceutics
journal-article
Conformational restrictions in ligand binding to the human intestinal di-/tripeptide transporter: implications for design of hPEPT1 targeted prodrugs.
journal-article
Conformational restrictions in ligand binding to the human intestinal di-/tripeptide transporter: Implications for design of hPEPT1 targeted prodrugs
Bioorganic and Medicinal Chemistry
journal-article
Conformational restrictions in ligand binding to the human intestinal di-/tripeptide transporter
Bioorganic & Medicinal Chemistry
journal-article
Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media.
journal-article
Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media
Molecular Pharmaceutics
journal-article
Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media
Molecular Pharmaceutics
journal-article
Forudsigelser med hjælp fra det virtuelle rum
Lægemiddelforskning
journal-article
Recent advances in therapeutic applications of human peptide transporters
Expert Opinion on Therapeutic Patents
journal-article
Recent advances in therapeutic applications of human transporters
Expert Opinion on Therapeutic Patents
journal-article
The F28Y substitution in the human intestinal di/tri-peptide transporter hPEPT1, causes altered pH-dependency of Gly-Sar transport
3rd World Conference on Drug Absorption, Transport and Delivery, Barcelona, Spain, 18/04/2005
conference-output
Genetic variants of the human H+/dipeptide transporter PEPT2: analysis of haplotype functions.
journal-article
Genetic variants of the human H+/dipeptide transporter PEPT2: Analysis of haplotype functions
Journal of Pharmacology and Experimental Therapeutics
journal-article
Genetic variants of the human H+/dipeptide transporter PEPT2
The Journal of Pharmacology and Experimental Therapeutics
journal-article
Dipeptidomimetic ketomethylene isosteres as pro-moieties for drug transport via the human intestinal di-/tripeptide transporter hPEPT1: design, synthesis, stability, and biological investigations.
journal-article
Dipeptidomimetic ketomethylene isosteres as pro-moieties for drug transport via the human intestinal di-/tripeptide transporter hPEPT1: Design, synthesis, stability, and biological investigations
Journal of Medicinal Chemistry
journal-article
Dipeptidomimetic ketomethylene isosteres as pro-moieties for drug transport via the human intestinal di-/tripeptide transporter hPEPT1
Journal of Medicinal Chemistry
journal-article
Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 cl.2.
journal-article
Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 c1.2
American Journal of Physiology - Renal Physiology
journal-article
Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 cl.2
American Journal of Physiology: Renal Physiology
journal-article
Phe-Gly dipeptidomimetics designed for the di-/tripeptide transporters PEPT1 and PEPT2: synthesis and biological investigations.
journal-article
Phe-Gly Dipeptidomimetics Designed for the Di-/Tripeptide Transporters PEPT1 and PEPT2: Synthesis and Biological Investigations
Journal of Medicinal Chemistry
journal-article
Phe-Gly dipeptidomimetics designed for the di-/tripeptide transporters PEPT1 and PEPT2
Journal of Medicinal Chemistry
journal-article
In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model.
journal-article
In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model
European Journal of Pharmaceutical Sciences
journal-article
In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model
European Journal of Pharmaceutical Sciences
journal-article
Intestinal solute carriers: an overview of trends and strategies for improving oral drug absorption.
journal-article
Intestinal solute carriers: An overview of trends and strategies for improving oral drug absorption
European Journal of Pharmaceutical Sciences
journal-article
Intestinal solute carriers
European Journal of Pharmaceutical Sciences
journal-article
Dipeptide ketomethylene isosteres as pro-moeities for drug transport via human intestinal di/tripeptide transport hPEPT1. Design, synthesis, stability and biological investigations
Journal of Medicinal Chemistry
journal-article
Di/tri-peptide transporters as drug delivery targets: regulation of transport under physiological and patho-physiological conditions.
journal-article
Erratum
Journal of Controlled Release
journal-article
Di/tri-peptide transporters as drug delivery targets: Regulation of transport under physiological and patho-physiological conditions
Current Drug Targets
journal-article
Di/tri-peptide transporters as drug delivery targets
Current Drug Targets
journal-article
Epidermal growth factor and insulin short-term increase hPepT1-mediated glycylsarcosine uptake in Caco-2 cells.
journal-article
Epidermal growth factor and insulin short-term increase hPepT1-mediated glycylsarcosine uptake in Caco-2 cells
Acta Physiologica Scandinavica
journal-article
Epidermal growth factor and insulin short-term increase hPEPT1-mediated glycylsarcosine uptake in Caco-2 cells
Acta Physiologica Scandinavica
journal-article
Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism.
journal-article
Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: Affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism
Journal of Controlled Release
journal-article
Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1
Journal of Controlled Release
journal-article
Erratum: Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: Affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism (Journal of Controlled Release (2003) 86 (279-292) PII: S0168365902004133)
Journal of Controlled Release
journal-article
Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line
Pharmaceutical Research
journal-article
Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line
Pharmaceutical Research
journal-article
Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1.
journal-article
Transport of peptidomimetic drugs by the intestinal di/tri-peptide transporter, PepT1
Pharmacology and Toxicology
journal-article
Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1
Basic & Clinical Pharmacology & Toxicology
journal-article
Human peptide transporters: Therapeutic applications
Expert Opinion on Therapeutic Patents
journal-article
Human peptide transporters
Expert Opinion on Therapeutic Patents
journal-article
Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line.
journal-article
Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line.
journal-article
Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line
Journal of Controlled Release
journal-article
Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line
Journal of Controlled Release
journal-article
Model prodrugs designed for the intestinal peptide transporter. A synthetic approach for coupling of hydroxy-containing compounds to dipeptides.
journal-article
Model prodrugs designed for the intestinal peptide transporter. A synthetic approach for coupling of hydroxy-containing compounds to dipeptides
European Journal of Pharmaceutical Sciences
journal-article
Model prodrugs designed for the intestinal peptide transporter
European Journal of Pharmaceutical Sciences
journal-article
Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line.
journal-article
Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line
American Journal of Physiology - Gastrointestinal and Liver Physiology
journal-article
Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line
American Journal of Physiology: Gastrointestinal and Liver Physiology
journal-article
Model prodrugs for the intestinal oligopeptide transporter: model drug release in aqueous solution and in various biological media.
journal-article
Model prodrugs for the intestinal oligopeptide transporter: Model drug release in aqueous solution and in various biological media
Journal of Controlled Release
journal-article
Model prodrugs for the intestinal oligopeptide transporter
Journal of Controlled Release
journal-article
Human proton/oligopeptide transporter (POT) genes: identification of putative human genes using bioinformatics.
journal-article
Human proton/oligopeptide transporter (POT) genes: identification of putative human genes using bioinformatics.
AAPS pharmSci [electronic resource]
journal-article
Human proton/oligopeptide transporter (POT) genes
AAPS PharmSci
journal-article